Disclaimer
CompoundIQ publishes research summaries for informational and educational purposes only. Nothing on this site constitutes medical advice, diagnosis, or treatment recommendations. Always consult a licensed healthcare provider. Many compounds listed are research chemicals not approved for human use.
GW-0742
GW-0742 is a highly selective PPARδ agonist structurally related to Cardarine (GW-501516). It is used in research settings to study PPARδ-mediated metabolic effects and has shown anti-inflammatory properties in preclinical studies.
Risk Level
High RiskDifficulty
Advanced| CAS Number | 317318-84-6 |
| Molecular Formula | C21H17F4NO3S2 |
| Class | Other |
| Category | Other Performance Compounds |
Mechanism of Action
GW-0742 selectively activates PPARδ with higher potency and selectivity than GW-501516. It regulates genes involved in fatty acid oxidation, inflammation, and glucose metabolism. It has demonstrated anti-inflammatory effects in skin and cardiovascular tissue in animal models.
Dosing Research
No human dosing data. Animal studies use 1-10 mg/kg. Research community references 10-20 mg/day based on extrapolation. No established protocols or cycle guidelines.
Side Effects & Risks
Shares the same PPARδ-related cancer concerns as GW-501516. No human safety data. Theoretical risks include metabolic disruption and unknown long-term effects. Should be considered high risk.
Research Studies
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Disclaimer
CompoundIQ publishes research summaries for informational and educational purposes only. Nothing on this site constitutes medical advice, diagnosis, or treatment recommendations. Always consult a licensed healthcare provider. Many compounds listed are research chemicals not approved for human use.